Method The target compound was synthesized from clarithromycin via hydrolyzation,acetylation,cyclic carbonatation,oxidation,decarbonatation,acylation,cyclic carbamatation and cyclization.
方法克拉霉素为起始原料,经水解、乙酰化、
碳
酯化、氧化、脱碳
酯化、酰化、
氨
酯化和
合等反应合成目标化合物。